ちょっとで大きな効果!
A potent seven-membered cyclic BTK (Bruton's tyrosine Kinase) chiral inhibitor conceived by structure-based drug design to lock its bioactive conformation - ScienceDirect https://t.co/46840Rw1Pi
ピペラジンからビシクロへの変換で物性改善!
Spirocyclic and Bicyclic 8-Nitrobenzothiazinones for Tuberculosis with Improved Physicochemical and Pharmacokinetic Properties https://t.co/O5Vv6ooxv4